Diane Boschelli: search on Z-Library

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1

Identification and optimization of indolo[2,3-c]quinoline inhibitors of IRAK4

Tumey, L. Nathan, Boschelli, Diane H., Bhagirath, Niala, Shim, Jaechul, Murphy, Elizabeth A., Goodwin, Deborah, Bennett, Eric M., Wang, Mengmeng, Lin, Lih-Ling, Press, Barry, Shen, Marina, Frisbie, Ri

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2014

Language:

english

File:

PDF, 2.40 MB

english, 2014

2

Optimization of 5-phenyl-3-pyridinecarbonitriles as PKCθ inhibitors

Diane H. Boschelli, Daniel Wang, Amar S. Prashad, Joan Subrath, Biqi Wu, Chuan Niu, Julie Lee, Xiaoke Yang, Agnes Brennan, Divya Chaudhary

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 318 KB

english, 2009

3

Synthesis of 2,6-di-tert-butylphenols linked to 1,3,4-oxadiazoles and 1,3,4-thiadiazoles

James B. Kramer, Diane H. Boschelli, David T. Connor

Journal:

Journal of Heterocyclic Chemistry

Year:

1994

File:

PDF, 439 KB

1994

4

Inhibition of Src Kinase Activity by 4-Anilino-7-thienyl-3-quinolinecarbonitriles.

Diane H. Boschelli, Daniel Y. Wang, Fei Ye, Ayako Yamashita, Nan Zhang, Dennis Powell, Jennifer Weber, Frank Boschelli

Journal:

Year:

2002

File:

PDF, 34 KB

2002

5

Inhibitors of Src tyrosine kinase: the preparation and structure–activity relationship of 4-anilino-3-cyanoquinolines and 4-anilinoquinazolines

Yanong D. Wang, Karen Miller, Diane H. Boschelli, Fei Ye, Biqi Wu, M.Brawner Floyd, Dennis W. Powell, Allan Wissner, Jennifer M. Weber, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 136 KB

english, 2000

6

Inhibition of Src kinase activity by 4-anilino-7-thienyl-3-quinolinecarbonitriles

Diane H. Boschelli, Daniel Y. Wang, Fei Ye, Ayako Yamashita, Nan Zhang, Dennis Powell, Jennifer Weber, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 133 KB

english, 2002

7

Synthesis and cyclooxygenase and 5-lipoxygenase inhibitory activity of some thiazolidene-4-one analogs of meclofenamic acid

Diane H. Boschelli, David T. Connor, Paul J. Kuipers, Clifford D. Wright

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1992

Language:

english

File:

PDF, 222 KB

english, 1992

8

Identification of 7-Phenylaminothieno- [3,2- b ]pyridine-6-carbonitriles as a New Class of Src Kinase Inhibitors

Boschelli, Diane H., Wu, Biqi, Barrios Sosa, Ana Carolina, Durutlic, Haris, Ye, Fei, Raifeld, Yuri, Golas, Jennifer M., Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 182 KB

english, 2004

9

Synthesis and PKCθ inhibitory activity of a series of 4-indolylamino-5-phenyl-3-pyridinecarbonitriles

Russell G. Dushin, Thomas Nittoli, Charles Ingalls, Diane H. Boschelli, Derek C. Cole, Allan Wissner, Julie Lee, Xiaoke Yang, Paul Morgan, Agnes Brennan, Divya Chaudhary

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 375 KB

english, 2009

10

Total synthesis of (±)-xanthocidin and (±)-desdihydroxy-4,5-dihydroxanthocidin

Diane Boschelli, Amos B. Smith III

Journal:

Tetrahedron Letters

Year:

1981

Language:

english

File:

PDF, 247 KB

english, 1981

11

Stereocontrolled total synthesis of (.+-.)-xanthocidin, two diastereomers, (.+-.)-epixanthocidin and (.+-.)-.beta.-isoxanthocidin, and (.+-.)-dedihydroxy-4,5-didehydroxanthocidin, a likely biosynthetic precursor

Smith, Amos B., Boschelli, Diane

Journal:

Journal of Organic Chemistry

Year:

1983

Language:

english

File:

PDF, 1.42 MB

english, 1983

12

Small Molecule Inhibitors of PKCθ as Potential Antiinflammatory Therapeutics

Boschelli, Diane

Journal:

Current Topics in Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 453 KB

english, 2009

13

ChemInform Abstract: Inhibitors of Src Tyrosine Kinase: The Preparation and Structure—Activity Relationship of 4-Anilino-3-cyanoquinolines and 4-Anilinoquinazolines.

Yanong D. Wang, Karen Miller, Diane H. Boschelli, Fei Ye, Biqi Wu, M. Brawner Floyd, Dennis W. Powell, Allan Wissner, Jennifer M. Weber, Frank Boschelli

Journal:

Year:

2001

File:

PDF, 33 KB

2001

14

Synthesis and Inhibition of Src Kinase Activity by 7-Ethenyl and 7-Ethynyl-4-anilino-3-quinolinecarbonitriles.

Ana Carolina Barrios Sosa, Diane H. Boschelli, Fei Ye, Jennifer M. Golas, Frank Boschelli

Journal:

Year:

2004

File:

PDF, 76 KB

2004

15

An asymmetric synthesis of (+)-kjellmanianone

Diane Boschelli, Amos B. Smith III, Orum D. Stringer, Robert H. Jenkins Jr., Franklin A. Davis

Journal:

Tetrahedron Letters

Year:

1981

Language:

english

File:

PDF, 265 KB

english, 1981

16

Crystal and molecular structure of geiparvarin

Bruce H. Toder, Diane Boschelli, Amos B. Smith

Journal:

Journal of Chemical Crystallography

Year:

1979

Language:

english

File:

PDF, 437 KB

english, 1979

17

A cell-based screen for inhibitors of protein folding and degradation

Frank Boschelli, Jennifer M. Golas, Roseann Petersen, Vincent Lau, Lei Chen, Diane Tkach, Qiang Zhao, Dave S. Fruhling, Hao Liu, Chaneun Nam, Kim T. Arndt

Journal:

Cell Stress and Chaperones

Year:

2010

Language:

english

File:

PDF, 518 KB

english, 2010

18

Structure−Activity Relationships for 1-Phenylbenzimidazoles as Selective ATP Site Inhibitors of the Platelet-Derived Growth Factor Receptor

Palmer, Brian D., Smaill, Jeff B., Boyd, Maruta, Boschelli, Diane H., Doherty, Annette M., Hamby, James M., Khatana, Sonya S., Kramer, James B., Kraker, Alan J., Panek, Robert L., Lu, Gina H., Dahring

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 169 KB

english, 1998

19

Synthesis and Src Kinase Inhibitory Activity of a Series of 4-Phenylamino-3-quinolinecarbonitriles

Boschelli, Diane H., Wang, Yanong D., Ye, Fei, Wu, Biqi, Zhang, Nan, Dutia, Minu, Powell, Dennis W., Wissner, Allan, Arndt, Kim, Weber, Jennifer M., Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 162 KB

english, 2001

20

Inhibition of Src kinase activity by 7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-heteroaryl-thieno[3,2-b]pyridine-6-carbonitriles

Diane H. Boschelli, Biqi Wu, Ana Carolina Barrios Sosa, Joan J. Chen, Jennifer M. Golas, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 113 KB

english, 2005

21

Synthesis of reversed hydroxamic acids of indomethacin: dual inhibitors of cyclooxygenase and 5-lipoxygenase

James B. Kramer, Diane H. Boschelli, David T. Connor, Catherine R. Kostlan, Daniel L. Flynn, Richard D. Dyer, Dirk A. Bornemeier, John A. Kennedy, Clifford D. Wright, Paul J. Kuipers

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1992

Language:

english

File:

PDF, 364 KB

english, 1992

22

Further Studies on Ethenyl and Ethynyl-4-phenylamino-3-quinolinecarbonitriles: Identification of a Subnanomolar Src Kinase Inhibitor.

Ana Carolina Barrios Sosa, Diane H. Boschelli, Biqi Wu, Yan Wang, Jennifer M. Golas

Journal:

Year:

2005

File:

PDF, 21 KB

2005

23

Preparation of a series of benzothieno[3,2-b]pyridine-3-carbonitriles and benzofuro[3,2-b]pyridine-3-carbonitriles

Diane H. Boschelli, Fei Ye

Journal:

Journal of Heterocyclic Chemistry

Year:

2002

Language:

english

File:

PDF, 74 KB

english, 2002

24

Inhibition of Src kinase activity by 7-ethynyl-4-phenylamino-3-quinolinecarbonitriles: Identification of SKS-927

Diane H. Boschelli, Ana Carolina Barrios Sosa, Jennifer M. Golas, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 150 KB

english, 2007

25

4-Anilino-7,8-dialkoxybenzo[ g ]quinoline-3-carbonitriles as Potent Src Kinase Inhibitors

Berger, Dan M., Dutia, Minu, Birnberg, Gary, Powell, Dennis, Boschelli, Diane H., Wang, Yanong D., Ravi, Malini, Yaczko, Deanna, Golas, Jennifer, Lucas, Judy, Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 576 KB

english, 2005

26

Preparation of a Series of Benzothieno[3,2-b]pyridine-3-carbonitriles and Benzofuro[3,2-b]pyridine-3-carbonitriles.

Diane H. Boschelli, Fei Ye

Journal:

Year:

2002

Language:

english

File:

PDF, 37 KB

english, 2002

27

Lead identification to generate isoquinolinedione inhibitors of insulin-like growth factor receptor (IGF-1R) for potential use in cancer treatment

Scott C. Mayer, Annette L. Banker, Frank Boschelli, Li Di, Mark Johnson, Cynthia Hess Kenny, Girija Krishnamurthy, Kristina Kutterer, Franklin Moy, Susan Petusky, Malini Ravi, Diane Tkach, Hwei-Ru Tso

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 273 KB

english, 2008

28

Enantioselective synthesis of (+)-kjellmanianone

Bang-Chi Chen, Michael C. Weismiller, Franklin A. Davis, Diane Boschelli, James R. Empfield, Amos B. Smith III

Journal:

Year:

1991

Language:

english

File:

PDF, 870 KB

english, 1991

29

Synthesis and Tyrosine Kinase Inhibitory Activity of a Series of 2-Amino-8H-pyrido[2,3-d]pyrimidines: Identification of Potent, Selective Platelet-Derived Growth Factor Receptor Tyrosine Kinase Inhibitors

Boschelli, Diane H., Wu, Zhipei, Klutchko, Sylvester R., Showalter, H. D. Hollis, Hamby, James M., Lu, Gina H., Major, Terry C., Dahring, Tawny K., Batley, Brian, Panek, Robert L.

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 219 KB

english, 1998

30

Synthesis and PKCθ inhibitory activity of a series of 4-(indol-5-ylamino)thieno[2,3-b]pyridine-5-carbonitriles

Diane H. Boschelli, Biqi Wu, Ana Carolina Barrios Sosa, Joan Chen, Magda Asselin, Derek C. Cole, Julie Lee, Xiaoke Yang, Divya Chaudhary

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 131 KB

english, 2008

31

A facile, scalable preparation of 4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carbonitriles

L. Nathan Tumey, Niala Bhagirath, Biqi Wu, Diane H. Boschelli

Journal:

Tetrahedron Letters

Year:

2008

Language:

english

File:

PDF, 161 KB

english, 2008

32

4-Anilino-6,7-dialkoxyquinoline-3-carbonitrile Inhibitors of Epidermal Growth Factor Receptor Kinase and Their Bioisosteric Relationship to the 4-Anilino-6,7-dialkoxyquinazoline Inhibitors

Wissner, Allan, Berger, Dan M., Boschelli, Diane H., Floyd, M. Brawner, Greenberger, Lee M., Gruber, Brian C., Johnson, Bernard D., Mamuya, Nellie, Nilakantan, Ramaswamy, Reich, Marvin F., Shen, Ru, T

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 384 KB

english, 2000

33

Synthesis and PKCθ inhibitory activity of a series of 5-vinyl phenyl sulfonamide-3-pyridinecarbonitriles

Jaechul Shim, Clark Eid, Julie Lee, Erica Liu, Divya Chaudhary, Diane H. Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 246 KB

english, 2009

34

Synthesis and evaluation of 4-Anilino-6,7-dialkoxy-3-quinolinecarbonitriles as inhibitors of kinases of the Ras-MAPK signaling cascade

Dan Berger, Minu Dutia, Dennis Powell, Biqi Wu, Allan Wissner, Diane H. Boschelli, M.Brawner Floyd, Nan Zhang, Nancy Torres, Jeremy Levin, Xuemei Du, Donald Wojciechowicz, Carolyn Discafani, Constance

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 173 KB

english, 2003

35

Synthesis and biological properties of 5,10-dideaza-5,6,7,8-tetrahydrofolic acid

Diane H. Boschelli, Stephanie Webber, John M. Whiteley, Arnold L. Oronsky, S.S. Kerwar

Journal:

Archives of Biochemistry and Biophysics

Year:

1988

Language:

english

File:

PDF, 554 KB

english, 1988

36

Editorial [ Hot Topic: Novel Medicinal Chemistry Approaches to New Anti-cancer Agents (Guest Editor: Diane H. Boschelli) ]

Boschelli, Diane

Journal:

Current Topics in Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 13 KB

english, 2008

37

C-5 Substituted heteroaryl 3-pyridinecarbonitriles as PKCθ inhibitors: Part I

Joan Subrath, Daniel Wang, Biqi Wu, Chuansheng Niu, Diane H. Boschelli, Julie Lee, Xiaoke Yang, Agnes Brennan, Divya Chaudhary

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 290 KB

english, 2009

38

Second generation 4-(4-methyl-1H-indol-5-ylamino)-2-phenylthieno[2,3-b]pyridine-5-carbonitrile PKCθ inhibitors

Biqi Wu, Diane H. Boschelli, Julie Lee, Xiaoke Yang, Divya Chaudhary

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 164 KB

english, 2009

39

7-(Aryl/heteroaryl-2-ylethynyl)-4-phenylamino-3-quinolinecarbonitriles as new Src kinase inhibitors: Addition of water solubilizing groups

Biqi Wu, Ana Carolina Barrios Sosa, Diane H. Boschelli, Frank Boschelli, Erick E. Honores, Jennifer M. Golas, Dennis W. Powell, Yanong D. Wang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 122 KB

english, 2006

40

Facile preparation of new 4-phenylamino-3-quinolinecarbonitrile Src kinase inhibitors via 7-fluoro intermediates: Identification of potent 7-amino analogs

Diane H. Boschelli, Biqi Wu, Fei Ye, Haris Durutlic, Jennifer M. Golas, Judy Lucas, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 172 KB

english, 2008

41

2-Substituted Aminopyrido[2,3-d]pyrimidin-7(8H)-ones. Structure−Activity Relationships Against Selected Tyrosine Kinases and in Vitro and in Vivo Anticancer Activity

Klutchko, Sylvester R., Hamby, James M., Boschelli, Diane H., Wu, Zhipei, Kraker, Alan J., Amar, Aneesa M., Hartl, Brian G., Shen, Cynthia, Klohs, Wayne D., Steinkampf, Randall W.

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 404 KB

english, 1998

42

Pyrido[2,3- d ]pyrimidin-7-one Inhibitors of Cyclin-Dependent Kinases

Barvian, Mark, Boschelli, Diane H., Cossrow, Jennifer, Dobrusin, Ellen, Fattaey, Ali, Fritsch, Alex, Fry, David, Harvey, Patricia, Keller, Paul, Garrett, Michelle, La, Frances, Leopold, Wilbur, McNama

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 228 KB

english, 2000

43

Cyclooxygenase and 5-lipoxygenase inhibitory activity of 2,6 di-t-butylphenols linked by a sulfur atom to 1,3,4-thiadiazoles and 1,3,4-oxadiazoles

James B. Kramer, Diane H. Boschelli, David T. Connor, Catherine R. Kostlan, Paul J. Kuipers, John A. Kennedy, Clifford D. Wright, Dirk A. Bornemeier, Richard D. Dyer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1993

Language:

english

File:

PDF, 240 KB

english, 1993

44

5-Vinyl-3-pyridinecarbonitrile inhibitors of PKCθ: Optimization of enzymatic and functional activity

L. Nathan Tumey, Niala Bhagirath, Agnes Brennan, Natasja Brooijmans, Julie Lee, Xiaoke Yang, Diane H. Boschelli

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 1.41 MB

english, 2009

45

Preparation of Benzothieno[2,3-f]-1,4-oxazepin- and -thiazepin-5(2H)-ones and of Benzothieno[3,2-e]-1,4-diazepin-5-ones

Khatana, Sonya S., Boschelli, Diane H., Kramer, James B., Connor, David T., Barth, Hubert, Stoss, Peter

Journal:

Journal of Organic Chemistry

Year:

1996

Language:

english

File:

PDF, 156 KB

english, 1996

46

Synthesis and Src Kinase Inhibitory Activity of 2-Phenyl- and 2-Thienyl-7-phenylaminothieno[3,2- b ]pyridine-6-carbonitriles

Boschelli, Diane H., Wu, Biqi, Barrios Sosa, Ana Carolina, Durutlic, Haris, Chen, Joan J., Wang, Yan, Golas, Jennifer M., Lucas, Judy, Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 197 KB

english, 2005

47

Pyrido[2,3- d ]pyrimidin-7-one Inhi-bitors of Cyclin-Dependent Kinases.

Barvian, Mark, Boschelli, Diane H., Cossrow, Jennifer, Dobrusin, Ellen, Fattaey, Ali, Fritsch, Alex, Fry, David, Harvey, Patricia, Keller, Paul, Garrett, Michelle, La, Frances, Leopold, Wilbur, McNama

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 15 KB

english, 2001

48

ChemInform Abstract: Synthesis and Src Kinase Inhibitory Activity of a Series of 4-Phenylamino-3-quinolinecarbonitriles.

Diane H. Boschelli, et al. et al.

Journal:

Year:

2001

Language:

english

File:

PDF, 30 KB

english, 2001

49

A facile one-pot synthesis of 2-substituted-3-aminoquinolines: preparation of benzo[b]naphthyridine-3-carbonitriles

Yanong D Wang, Diane H Boschelli, Steven Johnson, Erick Honores

Journal:

Year:

2004

Language:

english

File:

PDF, 296 KB

english, 2004

50

Synthesis of amphotericin B. 2. fragment C-D of the aglycone

Diane Boschelli, Toshiro Takemasa, Yasuhiro Nishitani, Satoru Masamune

Journal:

Tetrahedron Letters

Year:

1985

Language:

english

File:

PDF, 257 KB

english, 1985

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